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58

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T3036 Dydrogesterone

Progesterone Receptor Others
Dydrogesterone 是一种口服有效的孕激素,可作用于孕酮缺乏相关疾病。
T28362 PF-02413873

PF02413873

Progesterone Receptor Others
PF-02413873 是一种非甾体孕酮受体的竞争性拮抗剂,Ki 为 2.6 nM。 PF-02413873 可用于治疗子宫内膜异位症等妇科疾病的研究。
T13703 Gestonorone Capronate

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Gestonorone Capronate 是一种孕激素,在良性前列腺肥大和子宫内膜癌领域有研究价值。
T1514 Norethindrone

Norethisterone,炔诺酮

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Norethindrone (Norethisterone) 是孕激素,能够用于子宫内膜异位症、由激素水平异常引起的子宫出血和继发性闭经的研究。
T7537 Norgestimate

炔诺肟酯,诺孕酯

Progesterone Receptor Others
Norgestimate 是一种具有口服活性、高度选择性的孕激素活性和较小雄激素作用的孕激素,是一种合成的孕激素类似物。它可用作口服的避孕药。
T1596 Chlormadinone acetate

Gestafortin,醋酸氯地孕酮

Progesterone Receptor; Androgen Receptor Endocrinology/Hormones; Others
Chlormadinone acetate (Gestafortin) 是类固醇孕激素,具有抗雄激素和抗雌激素作用。
T8395 Nomegestrol acetate

Others; Progesterone Receptor Others
Nomegestrol acetate 是一种孕酮受体的完全激动剂,是一种高选择性孕激素。
T1541 Drospirenone

ZK 3059,屈螺酮,Dihydrospirorenone

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; COX Endocrinology/Hormones; Immunology/Inflammation; Neuroscience; Others
Drospirenone (ZK 3059) 是spironolactone 的类似物,是一种合成的孕酮。
T0996 Ethynodiol diacetate

Ethynodiol acetate,双醋炔诺醇,8080 CB

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Ethynodiol diacetate (Ethynodiol acetate) 是一种可用作激素避孕药的甾体孕激素,具有相对较少或没有雄激素效果,而具有显著雌激素作用。
T6819 Desogestrel

Org-2969,去氧孕烯,Desogen,Desogestrelum,Cerazette

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Desogestrel (Cerazette) 是第三代孕激素类似物,存在于许多口服避孕制剂中。
T6713 Ulipristal

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Ulipristal 是性孕酮受体 (progesterone receptor) 的选择性调节剂。它能够与孕激素受体结合,抑制 PR 介导的基因表达,降低生殖系统中孕激素的活性。
T5317 Cridanimod

CMA,吖啶酮乙酸,XBIO-101,10-carboxymethyl-9-acridanone

Progesterone Receptor; STING; IFNAR Immunology/Inflammation; Others
Cridanimod (10-carboxymethyl-9-acridanone, CMA) 是一种是小分子免疫调节剂和干扰素诱导剂,是一种孕酮受体激活剂,能够诱导 IFNα和IFNβ的表达,显著增加 PR 的表达。
T2577 Dienogest

地诺孕素,STS 557

Apoptosis; Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Others
Dienogest (STS 557) 是一种孕酮受体激动剂,作用于子宫内膜异位,有口服的子宫内膜活性。
T2527 Ulipristal acetate

Ulipristal,醋酸乌利司他,CDB-2914

Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy Autophagy; Endocrinology/Hormones; Others
Ulipristal acetate (CDB-2914) 是一种具有抗孕酮活性的选择性孕酮受体调节剂。它可抑制子宫平滑肌瘤病的生长。它通过抑制或延迟排卵和影响子宫内膜组织,可用作紧急避孕药。
T1490 Gestodene

SHB 331,WL 70,孕二烯酮

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Gestodene (WL 70) 是一种孕激素类避孕药。
T5174 Nestoron

醋酸烯诺孕酮,ST-1435,Segesterone Acetate,Nestorone,Elcometrine

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Nestoron (Segesterone Acetate) 是一种高度选择性和有效的孕激素,是一种 19-norprogesterone 衍生物,对progesterone receptors 具有高亲和力和选择性,可用作激素避孕药。
T14975 CJ-42794

CJ-042794

Others Others
CJ-42794 (CJ-042794)是前列腺素受体 EP4的选择性拮抗剂, 抑制[3H]-PGE2与 EP4受体结合的平均 pKi 为8.5, 对 EP4选择性比 EP1, EP2和 EP3高200多倍。
T0870 Altrenogest

R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Altrenogest (Allyltrenbolone) 是一种结构与trenbolone 相关的孕激素,能作用于孕激素受体。
T2231 Estradiol dipropionate

17-Beta-Estradiol-3,17-Dipropionate,3,17-二丙酸-17-BETA-雌二酯,二丙酸雌二醇

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) 是雌激素-孕激素的组合物,可用作雌激素 (estrogen) 孕激素 (progesterone) 激动剂。
T2567 Etonogestrel

3-Oxodesogestrel,3-keto-Desogestrel,依托孕烯,Nexplanon,Implanon

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Progesterone Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
Etonogestrel (Implanon) 是孕激素去氧孕烯的生物活性代谢物,与靶器官中的孕酮受体和雌激素受体高亲和力地结合,可诱导FKBP51mRNA 和蛋白表达。它是一种甾体孕激素,用作激素避孕药。
T1102 Mifepristone

C-1073,RU486,RU 38486,米非司酮

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; NO Synthase; Autophagy Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Others
Mifepristone (C-1073) 是一种黄体酮受体和糖皮质激素受体拮抗剂,在体外实验中的 IC50值分别为 0.2 nM 和 2.6 nM。
T20720 Norethisterone enanthate

NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564

Estrogen/progestogen Receptor Endocrinology/Hormones
Norethisterone enanthate (NSC-9564) 是一种口服有效的长效的孕激素。
T60056 Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl-

Progesterone Receptor Others
Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl- 是一种具有抗孕激素作用的孕酮受体拮抗剂。
T35054 Vilaprisan

BAY 1002670,BAY10-02670,BAY-1002670,BAY1002670,BAY-10-02670,BAY 10-02670

Progesterone Receptor Others
Vilaprisan (BAY 1002670) 是一种新型可口服且具有选择性的黄体酮受体调节剂 (SPRM),对子宫肌瘤 (UF) 具有抗增殖活性,可用于研究子宫肌瘤。
TP1862L [Sar9] Substance P acetate(77128-75-7 free base)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9] Substance P acetate(77128-75-7 free base) 是一种 NK-1 受体激动剂。 rNK1 特异性激动剂 [Sar-9,Met(O2)11]-SP 模拟了 SP 对孕酮代谢的作用。
T21395 Finerenone

BAY948862,BAY-948862,BAY94-8862,非奈利酮,BAY 94-8862,BAY-94-8862,BAY 948862

Glucocorticoid Receptor Endocrinology/Hormones
Finerenone (BAY-948862) 是一种选择性、具有口服活性的、非甾体类盐皮质激素受体拮抗剂 (IC50=18 nM)。与糖皮质激素受体、雄激素受体和孕酮受体相比,它表现出良好的选择性 (>500-fold)。它在心肾疾病研究中具有潜在的应用前景,如 2 型糖尿病和慢性肾脏疾病。
T16502 PF-3882845

Others Others
PF-3882845 also binds to the progesterone receptor (the binding IC50: 310 nM). PF-3882845 is a remarkably high affinity selective and orally efficacious mineralocorticoid receptor (MR binding IC50=2.7 nM) antagonist for hypertension and nephropathy.
T17291 ZK 216348

(+)-ZK 216348

Others Others
ZK 216348 also binds to Progesterone and mineralocorticoid receptors (IC50s: 20.4 nM and 79.9 nM, respectively). ZK 216348 is a nonsteroidal selective glucocorticoid receptor agonist (IC50: 20.3 nM). ZK 216348 has an anti-inflammatory activity similar to
T28995 Tosagestin

Org 30659,Org30659,Org-30659

Tosagestin is a progesterone receptor agonist.
T14332 Asoprisnil

J867

Others Others
Asoprisnil is a selective modulator of progesterone receptor.
T28263 Org-31710

Org 31710,Org31710

Org-31710 is a progesterone receptor antagonist potentially for contraception.
T29224 ZK112993

ZK-112993,ZK 112993

ZK112993 is an antagonist of human progesterone receptor.
T31082 CP-8668

UNII-5371O2R79D,CP 8668

CP-8668 is an orally active nonsteroidal progesterone receptor modulator with tetrahydrobenzoindolone skeleton.
T28264 Org-33628

Org-33628, a progesterone receptor antagonist, is used potentially for female contraception.
T27662 JNJ-1250132

JNJ 1250132,JNJ1250132

JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.
T27108 Cymipristone

ZXH951,ZXH 951,ZXH-951

Cymipristone, a progesterone receptor antagonist, is used potentially for termination of intrauterine pregnancy.
T34798 Telapristone

metabolite of telapristone acetate (CDB-4124)

Telapristone, is the active metabolite of telapristone acetate (also known as CDB-4124). Telapristone is a selective progesterone receptor modulator (SPRM) being studied for the treatment of certain progesterone-sensitive conditions.
T25304 Demegestone

R-2453,Lutionex,R 2453,RU 2453,R2453

Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat luteal insufficiency.
T28237 Onapristone

IVV-1001,ZK 98299,IVV 1001,ZK98299,ZK-98299,IVV1001

Onapristone, a progesterone receptor antagonist, is used potentially for the treatment of breast cancer, advanced prostate cancer, and inducer of vaginal bleeding.
T37319 5β-Dihydroprogesterone

5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP inhibits spontaneous contractions in isolated rat uterus when used at a concentration of 10 μg/ml, an effect that can be blocked by the progesterone receptor antagonist RU486 but not the GABAAreceptor antagonist picrotoxin .1It is a negative modulator of homooligomeric Ρ1 subunit-containing GABAAreceptors, inhibiting GABA-induced currents in...
T16985 Tanaproget

NSP-989

Others Others
Tanaproget is a novel nonsteroidal progesterone receptor agonist which can bind to the PR from various species with a higher relative affinity than reference steroidal progestins (IC50: 0.1 nM),
T19697 Norgestomet

SC21009,Norprogesterone, Syncro-Mate B,SC-21009,SC 21009

Norgestomet is a steroidal progestin of the 19-norprogesterone group used in veterinary medicine to control estrus and ovulation in cattle. In addition to the progesterone receptor, norgestomet possesses a weak (micromolar) affinity for the glucocorticoid
T28280 Oxendolone

Roxenone,Prostetin

Oxendolone is a steroidal progestin and antiandrogen. Oxendolone binds to the progesterone receptor (Ki = 20 nM) and androgen receptor (AR) (Ki = 320 nM) and acts as a weak but clinically relevant inhibitor of 5α-reductase.
T16396 OP-3633

Others Others
OP-3633 is an effective and selective steroidal glucocorticoid receptor (GR) antagonist (IC50: 29 nM). OP-3633 shows low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. It also has an inhibition of GR transcriptional activity.
T69895 Lonaprisan

Lonaprisan is an orally bioavailable pentafluoroethyl derivative of a mifepristone-related steroid with antiprogestagenic activity. Lonaprisan is a pure, highly receptor-selective progesterone receptor (PR) antagonist; binding of this agent to PRs inhibits PR activation and the associated proliferative effects. Unlike many other antiprogestins such as mifepristone, this agent does not appear to convert to an agonist in the presence of protein kinase A (PKA) activators and shows high antiprogesta...
T69717 Dimethandrolone

Dimethandrolone (DMA), also known by its developmental code name CDB-1321, is an experimental androgen/anabolic steroid (AAS) and progestogen medication which is under investigation for potential clinical use. Dimethandrolone is an AAS, and hence is an agonist of the androgen receptor, the biological target of androgens like testosterone. It is also a progestin, or a synthetic progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progestero...
T68473 WAY-255348

WAY-255348 is a potent nonsteroidal progesterone receptor (PR) antagonist. WAY-255348 inhibits the activity of progesterone. WAY-255348 achieves antagonist activity by binding to and subsequently preventing progesterone-induced nuclear accumulation, phosphorylation and promoter interactions of the PR. WAY-255348 bound PR conformation was similar to that of a progesterone agonist-bound PR and distinct from steroidal antagonist-bound PR conformations. WAY-255348 inhibits PR action through a novel ...
T26669 Asoprisnil ecamate

J956,J-956,J 956

Asoprisnil ecamate is a selective progesterone receptor modulator. Asoprisnil inhibits proliferation and induces apoptosis in cultured human uterine leiomyoma cells in the absence of comparable effects on myometrial cells. Asoprisnil inhibits embryo impla
T19684 Pregnanolone

SKF 6455,Kabi-2213,Kabi 2213,Eltanolone,Kabi2213,SKF6455

Pregnanolone is a cell membrane modulator potentially for the treatment of pain. Pregnanolone is an endogenous neurosteroid that is biosynthesized from progesterone. It is a positive allosteric modulator of the GABAA receptor, as well as a negative allost
T38448 (Rac)-Finerenone

(Rac)-Finerenone,(Rac)-BAY 94-8862

Rac-Finerenone, also known as (Rac)-BAY 94-8862, is the racemate derivative of Finerenone, a selective third-generation nonsteroidal mineralocorticoid receptor antagonist (MR) that is taken orally. With an IC50 value of 18 nM, Finerenone exhibits exceptional selectivity against the glucocorticoid receptor (GR), androgen receptor (AR), and progesterone receptor (>500-fold).

化合物

Dydrogesterone
Cat.No: T3036
Synonym:
Target: Progesterone Receptor
PF-02413873
Cat.No: T28362
Synonym: PF02413873
Target: Progesterone Receptor
Gestonorone Capronate
Cat.No: T13703
Synonym:
Target: Prostaglandin Receptor
Norethindrone
Cat.No: T1514
Synonym: Norethisterone,炔诺酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Norgestimate
Cat.No: T7537
Synonym: 炔诺肟酯,诺孕酯
Target: Progesterone Receptor
Chlormadinone acetate
Cat.No: T1596
Synonym: Gestafortin,醋酸氯地孕酮
Target: Progesterone Receptor, Androgen Receptor
Nomegestrol acetate
Cat.No: T8395
Synonym:
Target: Others, Progesterone Receptor
Drospirenone
Cat.No: T1541
Synonym: ZK 3059,屈螺酮,Dihydrospirorenone
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, COX
Ethynodiol diacetate
Cat.No: T0996
Synonym: Ethynodiol acetate,双醋炔诺醇,8080 CB
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Desogestrel
Cat.No: T6819
Synonym: Org-2969,去氧孕烯,Desogen,Desogestrelum,Cerazette
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Ulipristal
Cat.No: T6713
Synonym:
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Cridanimod
Cat.No: T5317
Synonym: CMA,吖啶酮乙酸,XBIO-101,10-carboxymethyl-9-acridanone
Target: Progesterone Receptor, STING, IFNAR
Dienogest
Cat.No: T2577
Synonym: 地诺孕素,STS 557
Target: Apoptosis, Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Ulipristal acetate
Cat.No: T2527
Synonym: Ulipristal,醋酸乌利司他,CDB-2914
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Gestodene
Cat.No: T1490
Synonym: SHB 331,WL 70,孕二烯酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Nestoron
Cat.No: T5174
Synonym: 醋酸烯诺孕酮,ST-1435,Segesterone Acetate,Nestorone,Elcometrine
Target: Estrogen/progestogen Receptor, Progesterone Receptor
CJ-42794
Cat.No: T14975
Synonym: CJ-042794
Target: Others
Altrenogest
Cat.No: T0870
Synonym: R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Estradiol dipropionate
Cat.No: T2231
Synonym: 17-Beta-Estradiol-3,17-Dipropionate,3,17-二丙酸-17-BETA-雌二酯,二丙酸雌二醇
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Progesterone Receptor
Etonogestrel
Cat.No: T2567
Synonym: 3-Oxodesogestrel,3-keto-Desogestrel,依托孕烯,Nexplanon,Implanon
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Mifepristone
Cat.No: T1102
Synonym: C-1073,RU486,RU 38486,米非司酮
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, NO Synthase, Autophagy
Norethisterone enanthate
Cat.No: T20720
Synonym: NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564
Target: Estrogen/progestogen Receptor
Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl-
Cat.No: T60056
Synonym:
Target: Progesterone Receptor
Vilaprisan
Cat.No: T35054
Synonym: BAY 1002670,BAY10-02670,BAY-1002670,BAY1002670,BAY-10-02670,BAY 10-02670
Target: Progesterone Receptor
[Sar9] Substance P acetate(77128-75-7 free base)
Cat.No: TP1862L
Synonym:
Target: Neurokinin receptor
Finerenone
Cat.No: T21395
Synonym: BAY948862,BAY-948862,BAY94-8862,非奈利酮,BAY 94-8862,BAY-94-8862,BAY 948862
Target: Glucocorticoid Receptor
PF-3882845
Cat.No: T16502
Synonym:
Target: Others
ZK 216348
Cat.No: T17291
Synonym: (+)-ZK 216348
Target: Others
Tosagestin
Cat.No: T28995
Synonym: Org 30659,Org30659,Org-30659
Target:
Asoprisnil
Cat.No: T14332
Synonym: J867
Target: Others
Org-31710
Cat.No: T28263
Synonym: Org 31710,Org31710
Target:
ZK112993
Cat.No: T29224
Synonym: ZK-112993,ZK 112993
Target:
CP-8668
Cat.No: T31082
Synonym: UNII-5371O2R79D,CP 8668
Target:
Org-33628
Cat.No: T28264
Synonym:
Target:
JNJ-1250132
Cat.No: T27662
Synonym: JNJ 1250132,JNJ1250132
Target:
Cymipristone
Cat.No: T27108
Synonym: ZXH951,ZXH 951,ZXH-951
Target:
Telapristone
Cat.No: T34798
Synonym: metabolite of telapristone acetate (CDB-4124)
Target:
Demegestone
Cat.No: T25304
Synonym: R-2453,Lutionex,R 2453,RU 2453,R2453
Target:
Onapristone
Cat.No: T28237
Synonym: IVV-1001,ZK 98299,IVV 1001,ZK98299,ZK-98299,IVV1001
Target:
5β-Dihydroprogesterone
Cat.No: T37319
Synonym:
Target:
Tanaproget
Cat.No: T16985
Synonym: NSP-989
Target: Others
Norgestomet
Cat.No: T19697
Synonym: SC21009,Norprogesterone, Syncro-Mate B,SC-21009,SC 21009
Target:
Oxendolone
Cat.No: T28280
Synonym: Roxenone,Prostetin
Target:
OP-3633
Cat.No: T16396
Synonym:
Target: Others
Lonaprisan
Cat.No: T69895
Synonym:
Target:
Dimethandrolone
Cat.No: T69717
Synonym:
Target:
WAY-255348
Cat.No: T68473
Synonym:
Target:
Asoprisnil ecamate
Cat.No: T26669
Synonym: J956,J-956,J 956
Target:
Pregnanolone
Cat.No: T19684
Synonym: SKF 6455,Kabi-2213,Kabi 2213,Eltanolone,Kabi2213,SKF6455
Target:
(Rac)-Finerenone
Cat.No: T38448
Synonym: (Rac)-Finerenone,(Rac)-BAY 94-8862
Target:
Cat. No. Product Name Target Signaling Pathways
T0478 Progesterone

孕酮,Pregn-4-ene-3,20-dione

Estrogen/progestogen Receptor; Progesterone Receptor; Opioid Receptor; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience; Others
Progesterone (Pregn-4-ene-3,20-dione) 是类固醇激素,能够调节月经周期。
T5040 Medroxyprogesterone

甲羟孕酮,甲孕酮

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Medroxyprogesterone 是一种合成的人孕酮变体,是孕酮受体激动剂,用于治疗肾癌。在兽医实践中用作发情调节剂。
T1263 Levonorgestrel

左炔诺孕酮,D-Norgestrel

Others; Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Levonorgestrel (D-Norgestrel) 是一种合成孕激素,可作用于孕酮受体。它是一种宫内节育器,可以抑制卵子受精。
T1261 Medroxyprogesterone Acetate

Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
Medroxyprogesterone Acetate (Farlutin) 是广泛使用的合成类固醇,与雄激素,孕酮及糖皮质激素受体均有作用。
T1284 Megestrol acetate

SC10363,醋酸甲地孕酮,BDH1298

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。
T1429 17α-Hydroxyprogesterone

Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮

Estrogen/progestogen Receptor; Progesterone Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
17α-Hydroxyprogesterone (17-OHP) 是一种内源性孕激素,其他类固醇激素(包括糖皮质激素,雌激素,和雄激素)生物合成的化学中间体。
T7974 Lynestrenol

Progesterone Receptor Others
Lynestrenol 是孕烷 X 受体 (PXR) 激动剂,能够作用于 hPXR(EC50:41 µM) 和 zfPXR(EC50:0.23 µM)。它是合成的孕酮,具有免疫刺激作用。
T7931 16a,17a-Epoxy-4-Pregnen-3,20-Dione

Others Others
16a,17a-Epoxy-4-Pregnen-3,20-Dione 是一种合成孕激素,是黄体酮激素的代谢产物,它通过与黄体酮受体结合发挥作用,已被用于研究孕激素对生殖器官的影响,激素对细胞生长和发育的影响,以及激素对免疫系统的影响。

天然产物

Progesterone
Cat.No: T0478
Synonym: 孕酮,Pregn-4-ene-3,20-dione
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite
Medroxyprogesterone
Cat.No: T5040
Synonym: 甲羟孕酮,甲孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Levonorgestrel
Cat.No: T1263
Synonym: 左炔诺孕酮,D-Norgestrel
Target: Others, Estrogen/progestogen Receptor, Progesterone Receptor
Medroxyprogesterone Acetate
Cat.No: T1261
Synonym: Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, Endogenous Metabolite
Megestrol acetate
Cat.No: T1284
Synonym: SC10363,醋酸甲地孕酮,BDH1298
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy
17α-Hydroxyprogesterone
Cat.No: T1429
Synonym: Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Lynestrenol
Cat.No: T7974
Synonym:
Target: Progesterone Receptor
16a,17a-Epoxy-4-Pregnen-3,20-Dione
Cat.No: T7931
Synonym:
Target: Others
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